115-137
Medicinal Chemistry of Neuronal Voltage-Gated Sodium Channel Blockers
138-144
A New Class of Symmetric Bisbenzimidazole-Based DNA Minor Groove-Binding Agents Showing Antitumor Activity
145-154
Estimation of Binding Affinities for HEPT and Nevirapine Analogues with HIV-1 Reverse Transcriptase via Monte Carlo Simulations
155-169
Synthesis and Comparative Molecular Field Analysis (CoMFA) of Symmetric and Nonsymmetric Cyclic Sulfamide HIV-1 Protease Inhibitors
170-179
2-Alkynyl-8-aryl-9-methyladenines as Novel Adenosine Receptor Antagonists: Their Synthesis and Structure-Activity Relationships toward Hepatic Glucose Production Induced via Agonism of the A2B Receptor
180-185
Cytotoxic Responses to Aromatic Ring and Configurational Variations in 
-Conidendrin, Podophyllotoxin, and Sikkimotoxin Derivatives
186-197
Synthesis and Structure-Activity Relationships of a New Model of Arylpiperazines. 5. Study of the Physicochemical Influence of the Pharmacophore on 5-HT1A/ 1-Adrenergic Receptor Affinity: Synthesis of a New Derivative with Mixed 5-HT1A/D2 Antagonist Properties
198-207
Synthesis and Structure-Activity Relationships of a New Model of Arylpiperazines. 6. Study of the 5-HT1A/ 1-Adrenergic Receptor Affinity by Classical Hansch Analysis, Artificial Neural Networks, and Computational Simulation of Ligand Recognition
208-214
Nucleosides and Nucleotides. 200. Reinvestigation of 5'-N-Ethylcarboxamidoadenosine Derivatives: Structure-Activity Relationships for P3 Purinoceptor-like Proteins
215-222
Synthesis and Characterization of Fluorescent and Photoactivatable MIP-1 Ligands and Interactions with Chemokine Receptors CCR1 and CCR5
223-231
Amino Acid Phosphoramidate Monoesters of 3'-Azido-3'-deoxythymidine: Relationship between Antiviral Potency and Intracellular Metabolism
232-244
Polyamine Analogue Antidiarrheals: A Structure-Activity Study
245-249
Dinuclear Alkyldiamine Platinum Antitumor Compounds: A Structure-Activity Relationship Study
250-260
Molecular Dynamics Study of the IIA Binding Site in Human Serum Albumin: Influence of the Protonation State of Lys195 and Lys199
261-268
Flavonolignan and Flavone Inhibitors of a Staphylococcus aureus Multidrug Resistance Pump: Structure-Activity Relationships
BRIEF ARTICLES
269-273
Crystal Structure of the Hydrated Strontium Salt of Methotrexate: Two Independent Molecules with Different Conformations
274-278
Agonist Activity at the Kinin B1 Receptor: Structural Requirements of the Central Tetrapeptide
BOOK REVIEWS
279-279
Membrane Structure in Disease and Drug Ther-apy Edited by Guido Zimmer. Marcel Dekker, New York. 2000. xxi + 530 pp. 15.5 × 23.5 cm. ISBN 0-8247-0361-8. $195.00.
279-279
ADDITIONS AND CORRECTIONS
280-280